VCP171
Catalogue number:
CAY30309-5 mg
Supplier:
Size:
5 mg
Product is available in:
£181.00
Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1018830-99-3
Purity:
≥98%
Formulation:
A crystalline solid
Molecular Weight:
347.4
Alternative Names:
[2-amino-4-[3-(trifluoromethyl)phenyl]-3-thienyl]phenyl-methanone
- Data sheet: View or download
- MSDS: View or download
Product Description:
A positive allosteric modulator of adenosine A1 receptors (EC50 = 15.8 µM in a kinetic assay measuring agonist dissociation); reduces AMPA receptor-mediated eEPSCs in lamina I and lamina II neurons in a rat model of neuropathic pain (EC50s = 1.995 and 0.251 µM, respectively) to a greater extent than in sham control animals (EC50s = 2.512 and 0.631 µM, respectively)
Storage Temperature:
-20°C