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Pantothenate Kinase Inhibitor

Catalogue number:
CAY31002-25 mg
Supplier:
Size:
25 mg _$$_
Product is available in:
  • UK
  • Ireland
  • Europe
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  • Rest of World
£535.00 Estimated delivery Fri 2 Aug
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

902614-04-4

Purity:

≥95%

Formulation:

A crystalline solid

Molecular Weight:

391.5

Alternative Names:

2,4-dimethyl-n-[3-(methylthio)phenyl]-pyrido[2′,3′:3,4]pyrazolo[1,5-a]pyrimidine-3-propanamide, pank inhibitor, panki

Product Description:

A reversible inhibitor of pantothenate kinase (PanK; IC50s = 70, 92, and 25 nM for PanK1β, PanK2, and PanK3, respectively); inhibits CoA biosynthesis in C3A cells (IC50 = 0.9 µM); sensitizes cells to ferroptosis inducers

Storage Temperature:

-20°C

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