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Centrinone

Catalogue number:
CAY24684-10 mg
Supplier:
Size:
10 mg
Product is available in:
  • UK
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£340.00 Estimated delivery Wed 7 Aug
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1798871-30-3

Purity:

≥95%

Formulation:

A solid

Molecular Weight:

633.6

Alternative Names:

2-[[2-fluoro-4-[[(2-fluoro-3-nitrophenyl)methyl]sulfonyl]phenyl]thio]-5-methoxy-n-(5-methyl-1h-pyrazol-3-yl)-6-(4-morpholinyl)-4-pyrimidinamine, lcr-263

Product Description:

A Plk4 inhibitor (Ki = 0.16 nM); >1,100- and >2,800-fold selective for Plk4 over Aurora A and Aurora B kinases, respectively, and a panel of 442 kinases at 100 nM; depletes centrosomes and induces apoptosis in HeLa cells at 125 nM

Storage Temperature:

-20°C

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