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PAP-1

Catalogue number:
CAY30105-10 mg
Supplier:
Size:
10 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£283.00 Estimated delivery Wed 7 Aug
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

870653-45-5

Purity:

≥98%

Formulation:

A solid

Molecular Weight:

350.4

Alternative Names:

4-(4-phenoxybutoxy)-7h-furo[3,2-g][1]benzopyran-7-one, 5-(4-phenoxybutoxy)psoralen

Product Description:

An inhibitor of Kv1.3 channels (EC50 = 2 nM at -80 mV in cells overexpressing the human channel); selective for Kv1.3 over a panel of 22 ion channels (EC50s = 45-15,000 nM for all); inhibits anti-CD3 antibody-induced proliferation of isolated human CCR7- effector memory T cells; inhibits ovalbumin-induced delayed-type hypersensitivity in rats at 3 mg/kg

Storage Temperature:

-20°C

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