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MK-5108

Catalogue number:
CAY19167-1 mg
Supplier:
Size:
1 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£74.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1010085-13-8

Purity:

≥95%

Formulation:

A crystalline solid

Molecular Weight:

461.9

Alternative Names:

trans-4-(3-chloro-2-fluorophenoxy)-1-[[6-(2-thiazolylamino)-2-pyridinyl]methyl]-cyclohexanecarboxylic acid, vx-689

Product Description:

A potent inhibitor of Aurora A (IC50 = 0.064 nM) that less potently inhibits Aurora B and Aurora C (IC50s =14 and 12 nM, respectively); blocks cell cycle progression and induces apoptosis in a diverse range of human tumor types; effective in vivo

Storage Temperature:

-20°C

CAY19167-1 mg: MK-5108
CAY19167-1 mg: MK-5108
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