PF-3758309
Catalogue number:
CAY19186-10 mg
Supplier:
Size:
10 mg
Product is available in:
£135.00
Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
898044-15-0
Purity:
≥98%
Formulation:
A crystalline solid
Molecular Weight:
490.6
Alternative Names:
n-[(1s)-2-(dimethylamino)-1-phenylethyl]-4,6-dihydro-6,6-dimethyl-3-[(2-methylthieno[3,2-d]pyrimidin-4-yl)amino]-pyrrolo[3,4-c]pyrazole-5(1h)-carboxamide, pf-309
- Data sheet: View or download
- MSDS: View or download
Product Description:
An ATP-competitive inhibitor of PAK4, preventing the phosphorylation of the PAK4 substrate GEF-H1 (IC50 = 1.3 nM) and blocking anchorage-independent growth of a panel of tumor cell lines (IC50 = 4.7 nM); blocks the growth of multiple human tumor xenografts
Storage Temperature:
-20°C
