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WZ4003

Catalogue number:
CAY19177-5 mg
Supplier:
Size:
5 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£130.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1214265-58-3

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

497

Alternative Names:

n-[3-[[5-chloro-2-[[2-methoxy-4-(4-methyl-1-piperazinyl)phenyl]amino]-4-pyrimidinyl]oxy]phenyl]-propanamide

Product Description:

A selective inhibitor of NUAK1 and NUAK2 (IC50s = 20 and 100 nM, respectively); inhibits the phosphorylation of the NUAK1 substrate MYPT1 at Ser445; inhibits proliferation and migration of mouse embryonic fibroblasts and U2OS cells at 10 µM in cell-based assays

Storage Temperature:

-20°C

CAY19177-5 mg: WZ4003
CAY19177-5 mg: WZ4003
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