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GNF-5837

Catalogue number:
CAY14883-5 mg
Supplier:
Size:
5 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£126.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1033769-28-6

Purity:

≥95%

Formulation:

A crystalline solid

Molecular Weight:

535.5

Alternative Names:

n-[3-[[2,3-dihydro-2-oxo-3-(1h-pyrrol-2-ylmethylene)-1h-indol-6-yl]amino]-4-methylphenyl]-n'-[2-fluoro-5-(trifluoromethyl)phenyl]-urea

Product Description:

A potent, bioavailable pan-Trk inhibitor that blocks the proliferation of cells expressing TEL-TrkA, TEL-TrkB, and TEL-TrkC (IC50s = 7, 9, and 11 nM, respectively); inhibits the growth of Ba/F3 and RIE cells expressing both TrkA and NGF with IC50 values of 42 and 17 nM, respectively

Storage Temperature:

-20°C

CAY14883-5 mg: GNF-5837
CAY14883-5 mg: GNF-5837
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