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AST-487

Catalogue number:
CAY19477-5 mg
Supplier:
Size:
5 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£146.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

630124-46-8

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

529.6

Alternative Names:

n-[4-[(4-ethyl-1-piperazinyl)methyl]-3-(trifluoromethyl)phenyl]-n'-[4-[[6-(methylamino)-4-pyrimidinyl]oxy]phenyl]-urea, nvp-ast-487

Product Description:

An inhibitor of RET (IC50 = 0.88 µM), FLT3 (Ki = 0.12 µM), KDR, c-Abl, and c-Kit; demonstrates antiproliferative activity in various cancer cells, including those with RET or FLT3 mutations

Storage Temperature:

-20°C

CAY19477-5 mg: AST-487
CAY19477-5 mg: AST-487
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