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MRT67307 (hydrochloride)

Catalogue number:
CAY19916-5 mg
Supplier:
Size:
5 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£167.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
Purity:

≥95%

Formulation:

A crystalline solid

Molecular Weight:

464.6

Alternative Names:

n-[3-[[5-cyclopropyl-2-[[3-(4-morpholinylmethyl)phenyl]amino]-4-pyrimidinyl]amino]propyl]-cyclobutanecarboxamide, hydrochloride

Product Description:

A kinase inhibitor that inhibits TBK1, MARK1-4, IKKε, and NUAK1 (IC50 values are 19, 27-52, 160, and 230 nM, respectively), SIKs (IC50s = 250, 67, and 430 nM for SIK1, SIK2, and SIK3, respectively) and ULK1 and ULK2 (IC50s = 45 and 38 nM, respectively)

Storage Temperature:

-20°C

CAY19916-5 mg: MRT67307
CAY19916-5 mg: MRT67307
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