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NVP-TNKS656

Catalogue number:
CAY19930-1 mg
Supplier:
Size:
1 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£130.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1419949-20-4

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

494.6

Alternative Names:

n-(cyclopropylmethyl)-4-(4-methoxybenzoyl)-n-[(3,5,7,8-tetrahydro-4-oxo-4h-pyrano[4,3-d]pyrimidin-2-yl)methyl]-1-piperidineacetamide

Product Description:

A TNKS2 inhibitor (IC50 = 6 nM); inhibits Wnt ligand-induced signaling in an HEK293 cell reporter assay (IC50 = 3.5 nM); reduces Axin 2 mRNA expression in MMTV-Wnt1 tumor bearing mice

Storage Temperature:

-20°C

CAY19930-1 mg: NVP-TNKS656
CAY19930-1 mg: NVP-TNKS656
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