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LY3214996

Catalogue number:
CAY27936-25 mg
Supplier:
Size:
25 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£1330.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1951483-29-6

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

453.6

Alternative Names:

5,6-dihydro-6,6-dimethyl-2-[2-[(1-methyl-1h-pyrazol-5-yl)amino]-4-pyrimidinyl]-5-[2-(4-morpholinyl)ethyl]-4h-thieno[2,3-c]pyrrol-4-one

Product Description:

An ERK1/2 inhibitor (IC50 = 5 nM for both); inhibits cell proliferation of tumor cells in vitro, including those expressing B-RAF, N-Ras, or K-Ras mutations in vitro; inhibits tumor growth in B-RAF or N-Ras mutant melanoma, B-RAF or K-Ras mutant colorectal, lung, and pancreatic cancer mouse xenograft models, as well as PDX mouse models

Storage Temperature:

-20°C

CAY27936-25 mg: LY3214996
CAY27936-25 mg: LY3214996
Details Cat number & supplier Size Price
LY3214996 CAY27936-10 mg · Cayman Chemical
CAY27936-10 mg
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LY3214996 CAY27936-5 mg · Cayman Chemical
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LY3214996 CAY27936-1 mg · Cayman Chemical
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Ara-G CAY27984-250 mg · Cayman Chemical
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MRX-2843 CAY27923-10 mg · Cayman Chemical
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Ara-G CAY27984-50 mg · Cayman Chemical
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