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XD14

Catalogue number:
CAY30740-25 mg
Supplier:
Size:
25 mg _$$_
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£601.00 Estimated delivery Fri 2 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1370888-71-3

Purity:

≥95%

Formulation:

A crystalline solid

Molecular Weight:

421.5

Alternative Names:

4-acetyl-n-[5-[(diethylamino)sulfonyl]-2-hydroxyphenyl]-3-ethyl-5-methyl-1h-pyrrole-2-carboxamide

Product Description:

A BRD inhibitor; binds to BRD2, -3, and 4 (Kds = 170, 380, and 160 nM); inhibits the growth of HL-60 cells (GI50 = ~20 µM), as well as various other cancer cells in vitro at 10 µM

Storage Temperature:

-20°C

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